Giclanfentrine
Giclanfentrine is a potent PDE3A inhibitor with an IC50 of 0.0058 μM. Giclanfentrine inhibits PDE4B1 activity with an IC50 of 12.9 μM. Giclanfentrine is applicable to studies related to PDE3/cAMP signaling.
For research use only. We do not sell to patients.
- CAS No.: 2408152-69-0
- Formula: C30H35N7O5
- Molecular Weight:573.64
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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PDE3A 0.0058 μM (IC50) |
PDE4B1 12.9 μM (IC50) |
Chemical Information
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CAS No. 2408152-69-0
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Molecular Weight 573.64
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Formula C30H35N7O5
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SMILES
O=C(C1=C(N=NN1C)O)NCCN2/C(C=C3C4=C(CCN3C2=O)C=C(OCC)C(OC)=C4)=N/C5=C(C)C=C(C)C=C5C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)