PD-334581
Based on 1 Customer Validation
PD-334581 is a MEK1 inhibitor.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 99.72%
- CAS 番号: 548756-68-9
- 分子式: C20H19F3IN5O2
- 分子量:545.30
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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MEK アイソフォーム固有の製品をすべて表示
More
生物活性
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MEK1 |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| Colon 26 | IC50 |
0.032 M
Compound: 12J
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Inhibition of MEK in mouse Colon 26 cells by Western blot
Inhibition of MEK in mouse Colon 26 cells by Western blot
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[PMID: 18951019] |
化学情報
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CAS 番号 548756-68-9
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性状 Solid
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分子量 545.30
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分子式 C20H19F3IN5O2
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Color White to yellow
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SMILES
FC1=C(F)C(NC2=CC=C(C=C2F)I)=C(C3=NN=C(NCCN4CCOCC4)O3)C=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 12.5 mg/mL (22.92 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (272 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.8339 mL | 9.1693 mL | 18.3385 mL | 45.8463 mL |
| 5 mM | 0.3668 mL | 1.8339 mL | 3.6677 mL | 9.1693 mL | |
| 10 mM | 0.1834 mL | 0.9169 mL | 1.8339 mL | 4.5846 mL | |
| 15 mM | 0.1223 mL | 0.6113 mL | 1.2226 mL | 3.0564 mL | |
| 20 mM | 0.0917 mL | 0.4585 mL | 0.9169 mL | 2.2923 mL |
PD-334581 関連分類
HY-107619 関連分類
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