PSB-1901
Based on 1 Customer Validation
PSB-1901 is a potent A2B adenosine receptor (A2BAR) antagonist with Kis of 0.0835 nM and 0.131 nM for human and mouse A2BARs respectively. PSB-1901 can be used for the research of cancer.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度 : 96.33%
- CAS 番号: 2332835-02-4
- 分子式: C24H25BrN6O4S
- 分子量:573.46
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
Adenosine Receptor アイソフォーム固有の製品をすべて表示
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生物活性
製品説明
IC50 & Target
Ki: 0.0835 nM (human A2BAR), 0.131 nM (mouse A2BAR)[1]
化学情報
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CAS 番号 2332835-02-4
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性状 Solid
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分子量 573.46
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分子式 C24H25BrN6O4S
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Color White to off-white
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SMILES
O=C1NC2=C(C(N1CCC)=O)NC(C3=CC=C(S(=O)(N4CCN(CC4)C5=CC=C(C=C5)Br)=O)C=C3)=N2
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
体外:
DMSO : ≥ 100 mg/mL (174.38 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (268 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.7438 mL | 8.7190 mL | 17.4380 mL | 43.5950 mL |
| 5 mM | 0.3488 mL | 1.7438 mL | 3.4876 mL | 8.7190 mL | |
| 10 mM | 0.1744 mL | 0.8719 mL | 1.7438 mL | 4.3595 mL | |
| 15 mM | 0.1163 mL | 0.5813 mL | 1.1625 mL | 2.9063 mL | |
| 20 mM | 0.0872 mL | 0.4360 mL | 0.8719 mL | 2.1798 mL | |
| 25 mM | 0.0698 mL | 0.3488 mL | 0.6975 mL | 1.7438 mL | |
| 30 mM | 0.0581 mL | 0.2906 mL | 0.5813 mL | 1.4532 mL | |
| 40 mM | 0.0436 mL | 0.2180 mL | 0.4360 mL | 1.0899 mL | |
| 50 mM | 0.0349 mL | 0.1744 mL | 0.3488 mL | 0.8719 mL | |
| 60 mM | 0.0291 mL | 0.1453 mL | 0.2906 mL | 0.7266 mL | |
| 80 mM | 0.0218 mL | 0.1090 mL | 0.2180 mL | 0.5449 mL | |
| 100 mM | 0.0174 mL | 0.0872 mL | 0.1744 mL | 0.4360 mL |
PSB-1901 関連分類
HY-153897 関連分類
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