KAT6-IN-4
KAT6-IN-4 (Compound Example 2) is a selective lysine acetyltransferase 6 (KAT6) inhibitor. KAT6-IN-4 suppresses transcription of oncogenes like ERα. KAT6-IN-4 demonstrates potent antitumor efficacy in ER+/HER2- breast cancer xenografts. KAT6-IN-4 is promising for research of KAT6-driven malignancies (e.g., breast cancer, NSCLC).
For research use only. We do not sell to patients.
- CAS No.: 2901797-38-2
- Formula: C22H22N4O6S
- Molecular Weight:470.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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ERα |
Chemical Information
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CAS No. 2901797-38-2
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Molecular Weight 470.50
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Formula C22H22N4O6S
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SMILES
O=S(NC1=NOC2=CC(CN3N=CC=C3)=C4C(OCCC4)=C21)(C5=C(OC)C=CC=C5OC)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)