1. Membrane Transporter/Ion Channel
  2. Sodium Channel
  3. (R)-Funapide

(R)-Funapide (Synonyms: (R)-TV 45070; (R)-XEN402)

Cat. No.: HY-16723A
Handling Instructions

(R)-Funapide ((R)-TV 45070) is the less active R-enantiomer of Funapide. Funapide is a potent Nav1.7 sodium channel blocker that can be used for pain research.

For research use only. We do not sell to patients.

(R)-Funapide Chemical Structure

(R)-Funapide Chemical Structure

CAS No. : 1259933-15-7

Size Price Stock Quantity
5 mg USD 480 In-stock
Estimated Time of Arrival: December 31
10 mg USD 800 In-stock
Estimated Time of Arrival: December 31
25 mg USD 1650 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
100 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of (R)-Funapide:

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Description

(R)-Funapide ((R)-TV 45070) is the less active R-enantiomer of Funapide. Funapide is a potent Nav1.7 sodium channel blocker that can be used for pain research[1].

Molecular Weight

429.35

Formula

C₂₂H₁₄F₃NO₅

CAS No.
SMILES

O=C([[email protected]@]12COC3=C1C=C(OCO4)C4=C3)N(CC5=CC=C(C(F)(F)F)O5)C6=C2C=CC=C6

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 220 mg/mL (512.40 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.3291 mL 11.6455 mL 23.2910 mL
5 mM 0.4658 mL 2.3291 mL 4.6582 mL
10 mM 0.2329 mL 1.1646 mL 2.3291 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: 5 mg/mL (11.65 mM); Suspended solution; Need ultrasonic

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: 5 mg/mL (11.65 mM); Suspended solution; Need ultrasonic

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 5 mg/mL (11.65 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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  • Molarity Calculator

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This equation is commonly abbreviated as: C1V1 = C2V2

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Keywords:

(R)-Funapide(R)-TV 45070 (R)-XEN402Sodium ChannelNa channelsNa+ channelsNav1.7painInhibitorinhibitorinhibit

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Product Name:
(R)-Funapide
Cat. No.:
HY-16723A
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