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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
33 Results for "
β-adrenoceptor antagonist
" in MedChemExpress (MCE) Product Catalog:
Products (33)
33 Results for "β-adrenoceptor antagonist" in MCE Product Catalog:
9
9 Publications Verification
Cat. No.: HY-B1517
CAS No.: 13655-52-2
Synonyms: (RS)-Alprenolol; dl-Alprenolol
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Alprenolol ((RS)-Alprenolol; dl-Alprenolol) is an orally active non-selective β-adrenoceptor antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .
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9 Publications Verification
Cat. No.: HY-B1517A
CAS No.: 13707-88-5
Synonyms: (RS)-Alprenolol hydrochloride; dl-Alprenolol hydrochloride
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Alprenolol ((RS)-Alprenolol; dl-Alprenolol) hydrochloride is an orally active non-selective β-adrenoceptor antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol hydrochloride is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .
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1 Cited Publications
Cat. No.: HY-A0295
CAS No.: 13071-11-9
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(R)-Propranolol hydrochloride is a less active enantiomer of the β-adrenoceptor antagonist propranolol (HY-B0573). Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively .
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Penbutolol sulfate ((-)-Terbuclomine) is a potent β-adrenoceptor and 5-HT receptor antagonist with Ki of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3 .
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1 Cited Publications
Cat. No.: HY-116790
CAS No.: 38363-40-5
Synonyms: (S)-Penbutolol; (-)-Isopenbutolol
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(-)-Penbutolol ((S)-Penbutolol) is a potent β-adrenoceptor and 5-HT receptor antagonist with Ki values of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3 .
Synonyms: (-)-Pindolol; (S)-(-)-Pindolol; l-Pindolol
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Espindolol ((-)-pindolol) is a reversible, competitive and orally active 5-HT1A/1B antagonist. lEspindolol is a partial β-adrenoceptor agonist. Espindolol can be used for the research of neurological disease .
Synonyms: (R)-Penbutolol; (+)-Isopenbutolol
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(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC50 of 0.74 μM . (+)-Penbutolol is an optical isomer of l-penbutolol with Na + channel-blocking action .
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VK-II-86 is a Carvedilol (HY-B0006) analogue lacking antagonist activity at β-adrenoceptors, in hypokalaemia. VK-II-86 prevents hypokalaemia-induced ventricular arrhythmia through multi-channel effects. VK-II-86 prevents all hypokalaemia-induced changes in ion channel activity and oxidative stress .
Cat. No.: HY-B1562B
CAS No.: 82857-38-3
Synonyms: (±)-Bopindolol malonate
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Bopindolol ((±)-Bopindolol) malonate is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity. Bopindolol malonate is non-selective for β1- and β2-ARs and has low affinity for β3-AR subtype. Bopindolol malonate has intrinsic sympathomimetic as well as membrane stabilizing actions, inhibits renin secretion, and interacts with 5-HT receptors. Bopindolol malonate is a proagent of Pindolol (HY-B0982). Bopindolol malonate can be used for essential and renovascular hypertension research.
Cat. No.: HY-A0252
CAS No.: 14556-46-8
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Bupranolol is an orally active, competitive and non-selective β-adrenoceptor antagonist without intrinsic sympathomimetic activity .
Cat. No.: HY-A0252R
CAS No.: 14556-46-8
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Bupranolol (Standard) is the analytical standard of Bupranolol. This product is intended for research and analytical applications. Bupranolol is an orally active, competitive and non-selective β-adrenoceptor antagonist without intrinsic sympathomimetic activity .
Cat. No.: HY-B1517AR
CAS No.: 13707-88-5
Synonyms: (RS)-Alprenolol hydrochloride (Standard); dl-Alprenolol hydrochloride (Standard)
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Alprenolol (hydrochloride) (Standard) is the analytical standard of Alprenolol (hydrochloride). This product is intended for research and analytical applications. Alprenolol ((RS)-Alprenolol; dl-Alprenolol) hydrochloride is an orally active non-selective β-adrenoceptor antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol hydrochloride is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .
Cat. No.: HY-19578B
CAS No.: 874882-92-5
Synonyms: (±)-Isamoltane hemifumarate
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Isamoltane hemifumarate is a selective antagonist of 5-HT1B receptor, with an IC50 of 39 nM for inhibits the binding of [ 125I]ICYP to 5-HT1B recognition sites in rat brain membranes. Isamoltane hemifumarate is also a β-adrenoceptor ligand, with an IC50 of 8.4 nM. Isamoltane hemifumarate shows anxiolytic activity .
Cat. No.: HY-17495
CAS No.: 51781-06-7
Synonyms: OPC-1085
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Carteolol is a non-selective β-adrenoceptor antagonist. Carteolol induces apoptosis via a caspase activated and mitochondrial-dependent pathway. Carteolol can be used for glaucoma research .
Cat. No.: HY-B1517B
CAS No.: 67824-72-0
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Alprenolol benzoate is an orally active non-selective β-adrenoceptor antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol benzoate is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .
Cat. No.: HY-U00019
CAS No.: 59110-35-9
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Pamatolol is a cardioselective beta-adrenoceptor antagonist without sympathomimetic activity.
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Labetalone hydrochloride is an impurity of Labetalol. Labetalol is an orally active adrenoceptor blocking agent which is a competitive antagonist at both alpha- and beta-adrenoceptor sites .
Cat. No.: HY-P1376
CAS No.: 143675-79-0
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Cat. No.: HY-121692A
CAS No.: 16768-36-8
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(S)-Alprenolol is a potent and nonselective β-adrenoceptor antagonist .
Cat. No.: HY-106499
CAS No.: 66264-77-5
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Sulfinalol is an orally active β-adrenoceptor antagonist with direct vasodilator activity .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
