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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
143 Results for "
EphA
" in MedChemExpress (MCE) Product Catalog:
Products (143)
143 Results for "EphA" in MCE Product Catalog:
9
9 Publications Verification
Synonyms: BHG712
Target:
Domaines de recherche:
NVP-BHG712 is an oral active EphB4 kinase autophosphorylation inhibitor, with IC50 values of 3.3 nM and 3.0 nM for EphA2 and EphB4, respectively .
3
3 Cited Publications
Cat. No.: HY-P2264
CAS No.: 676657-00-4
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2
2 Cited Publications
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Domaines de recherche:
NVP-BHG712 isomer, a regioisomer of NVP-BHG712, shows conserved non-bonded binding to EPHA2 and EPHB4 .
2
Category:
Uncaria rhynchophylla (Miq.) Miq. ex Havil. Alkaloids Other Diseases Rubiaceae Plants Disease Research Fields Indole Alkaloids
Target:
1
1
1 Cited Publications
Cat. No.: HY-P10579
CAS No.: 2225868-19-7
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Domaines de recherche:
1
1 Cited Publications
Cat. No.: HY-P0177
CAS No.: 2034159-30-1
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1
Category:
Human Gut Microbiota Metabolites Microorganisms Neurological Disease Ketones, Aldehydes, Acids Endogenous metabolite Disease Research Fields Inflammation/Immunology
Target:
Target:
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EphA2 agonist 1 (Compound 7bg) is a potent EphA2 receptor agonist. EphA2 agonist 1 shows great potency and selectivity toward EphA2 overexpressed glioblastoma cells and stimulates EphA2 phosphorylation .
Cat. No.: HY-169849
CAS No.: 1428095-28-6
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Domaines de recherche:
EphA2 antagonist 1 (4b) is a bile acid conjugate and an ephrin type-A receptor 2 (EPHA2) inhibitor .
Cat. No.: HY-W078239
CAS No.: 313701-92-7
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Domaines de recherche:
EPHA4 antagonist-1 (Compound 2) is an EphA4 receptor antagonist. EPHA4 antagonist-1 is also an EphA2 receptor antagonist. EPHA4 antagonist-1 inhibits ephrin-A5 AP binding to EphA4 Fc receptor, with an IC50 of 10 μM .
Cat. No.: HY-159174
Domaines de recherche:
EPHA2/A4/GAK-IN-1 (compound 55) is a potent inhibitor of EPHA2/EPHA4 and GAK with KD values of 180.5 nM for EPHA2 and 19.2 nM for GAK, respectively. EPHA2/GAK-IN-1 shows an extrapolated half-life time of 4.6 h in a microsomal stability assay. EPHA2/GAK-IN-1 shows antiviral activity and prevents dengue virus infection of Huh7 liver cells .
Cat. No.: HY-146141
CAS No.: 2169273-66-7
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EphA2 agonist 2 (Lead compound) is a selective EphA2 agonist with antitumor activities. EphA2 agonist 2 can cross the BBB .
Cat. No.: HY-P11243
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Cat. No.: HY-RS04424
Target:
Domaines de recherche:
EPHA1 Human Pre-designed siRNA Set A contains three designed siRNAs for EPHA1 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS04425
Target:
Domaines de recherche:
EPHA10 Human Pre-designed siRNA Set A contains three designed siRNAs for EPHA10 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS04426
Target:
Domaines de recherche:
EPHA2 Human Pre-designed siRNA Set A contains three designed siRNAs for EPHA2 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS04427
Target:
Domaines de recherche:
EPHA3 Human Pre-designed siRNA Set A contains three designed siRNAs for EPHA3 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS04428
Target:
Domaines de recherche:
EPHA4 Human Pre-designed siRNA Set A contains three designed siRNAs for EPHA4 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-RS04429
Target:
Domaines de recherche:
EPHA5 Human Pre-designed siRNA Set A contains three designed siRNAs for EPHA5 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
