SmCB1-IN-1
SmCB1-IN-1 (Compound 2h) is an inhibitor for S. mansoni cathepsin B1 (SmCB1) with an Ki of 0.05 μM. SmCB1-IN-1 exhibits selectivity toward human off-target cathepsins (29% and 37% inhibition for CatB and CatL at 20 μM). SmCB1-IN-1 inhibits 68% Schistosoma mansoni at 1 μM.
For research use only. We do not sell to patients.
- Formula: C26H25NO6S
- Molecular Weight:479.54
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Schistosome |
S. mansoni cathepsin B1 0.05 μM (IC50) |
Chemical Information
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Molecular Weight 479.54
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Formula C26H25NO6S
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SMILES
O=S(/C=C/[C@@H](NC(C1=C2C(OCCO2)=CC=C1)=O)CCC3=CC=CC=C3)(OC4=CC=CC=C4)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)