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BI-3802 

Cat. No.: HY-108705
Handling Instructions

BI-3802 is a highly potent BCL6 degrader, inhibiting the BTB domain of BCL6, with an IC50 of ≤3 nM; BI-3802 has antitumor activity.

For research use only. We do not sell to patients.

BI-3802 Chemical Structure

BI-3802 Chemical Structure

CAS No. : 2166387-65-9

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

BI-3802 is a highly potent BCL6 degrader, inhibiting the BTB domain of BCL6, with an IC50 of ≤3 nM; BI-3802 has antitumor activity.

IC50 & Target

IC50: ≤3 nM (BCL6 BTB)[1]

In Vitro

BI-3802 is a BCL6 inhibitor, with an IC50 of ≤3 nM. BI-3802 shows an IC50 of 43 nM for the cellular BCL6[1].

Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0619 mL 10.3097 mL 20.6194 mL
5 mM 0.4124 mL 2.0619 mL 4.1239 mL
10 mM 0.2062 mL 1.0310 mL 2.0619 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

484.98

Formula

C₂₄H₂₉ClN₆O₃

CAS No.

2166387-65-9

SMILES

ClC1=CN=C(N2C[[email protected]](C)C[[email protected]](C)C2)N=C1NC3=CC(C=C(OCC(NC)=O)C(N4C)=O)=C4C=C3

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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Product Name:
BI-3802
Cat. No.:
HY-108705
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BI-3802

Cat. No.: HY-108705