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BI-3802

3 Cited Publications
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Based on 3 publication(s) in Google Scholar

BI-3802, a chemical probe, is a highly potent BCL6 degrader and inhibits the Bric-à-brac (BTB) domain of BCL6 with an IC50 of ≤3 nM. BI-3802 induces the polymerization of BCL6 and promotes BCL6 degration depended on E3 ligase SIAH1. BI-3802 has antitumor activity.

Para uso exclusivo en investigación. No vendemos a pacientes.

The BI-3802 was designed by Boehringer Ingelheim and could be obtained free of charge through the Boehringer Ingelheim open innovation portal opnMe.com, associated with its negative control.

  • Pureza: 99.27%
  • No. CAS: 2166387-65-9
  • Fòrmula: C24H29ClN6O3
  • Peso molecular:484.98
  • Almacenamiento:
    Powder   -20°C, 3 years , 4°C, 2 years ; In solvent   -80°C, 6 months , -20°C, 1 month
  • BI-3802 Chemical Structure
    BI-3802 Chemical Structure
  • Experimental Validation Results for BI-3802
  • Experimental Validation Results for BI-3802
No. CAS: 2166387-65-9
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Encuentre su distribuidor local Your local distributor: Hycultec GmbHHycultec
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Bio/Physico-chemical AssayCell Imaging/Staining
  • Bio/Physico-chemical Assay
  • Cell Imaging/Staining

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  • BI-3802 Chemical Structure
    BI-3802 Chemical Structure
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  • 1/16

    BI-3802 purchased from MedChemExpress. Usage Cited in: Genome Biol. 2025 Sep 2;26(1):264. [Abstract]

    Customer Validation
     Terminal cumulative MSD of NONO-GFP foci at final time point. Each circle indicates a single NONO-GFP focus. For untransfected groups, 45 foci were analyzed from 10 cells; for + BI-3802, 38 from 15 cells; and for + BI-3812, 37 foci from 15 cells across three biological replicates.

  • 1/16

    BI-3802 purchased from MedChemExpress. Usage Cited in: Genome Biol. 2025 Sep 2;26(1):264. [Abstract]

    Customer Validation
     Compared to cells untransfected with the inducible HP1α switch, both the length of trajectories and terminal MSD of NONO-GFP foci were increased by the promoted condensation of HP1α using BI-3802 (1 μM).

  • BI-3802