1. Metabolic Enzyme/Protease
  2. Phosphatase

Rilapladib (Synonyms: SB 659032)

Cat. No.: HY-102004
Handling Instructions

Rilapladib is a selective Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) inhibitor with an IC50 of 230 pM.

For research use only. We do not sell to patients.

Rilapladib Chemical Structure

Rilapladib Chemical Structure

CAS No. : 412950-08-4

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  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Rilapladib is a selective Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) inhibitor with an IC50 of 230 pM.

IC50 & Target

IC50: 230 pM (Lp-PLA2)[1].

Clinical Trial
Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.3590 mL 6.7952 mL 13.5905 mL
5 mM 0.2718 mL 1.3590 mL 2.7181 mL
10 mM 0.1359 mL 0.6795 mL 1.3590 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

735.81

Formula

C₄₀H₃₈F₅N₃O₃S

CAS No.

412950-08-4

SMILES

O=C(N(C1CCN(CCOC)CC1)CC2=CC=C(C3=CC=C(C(F)(F)F)C=C3)C=C2)CN4C(SCC5=CC=CC(F)=C5F)=CC(C6=C4C=CC=C6)=O

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Rilapladib
Cat. No.:
HY-102004
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Rilapladib

Cat. No.: HY-102004