Tenalisib R Enantiomer
Based on 1 Customer Validation
Tenalisib R Enantiomer (RP6530 R Enantiomer) is an R enantiomer of Tenalisib. Tenalisib is a potent and selective PI3Kδ and PI3Kγ inhibitor with IC50 values of 25 and 33 nM, respectively.
For research use only. We do not sell to patients.
- Purity: 99.63%
- CAS No.: 1639417-54-1
- Formula: C23H18FN5O2
- Molecular Weight:415.42
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Biological Activity
Chemical Information
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CAS No. 1639417-54-1
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Appearance Solid
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Molecular Weight 415.42
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Formula C23H18FN5O2
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Color White to off-white
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SMILES
O=C1C(C2=CC=CC(F)=C2)=C([C@H](NC3=C4N=CNC4=NC=N3)CC)OC5=CC=CC=C15
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Synonyms
RP6530 R Enantiomer
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
DMSO : 100 mg/mL (240.72 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (277 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.4072 mL | 12.0360 mL | 24.0720 mL | 60.1801 mL |
| 5 mM | 0.4814 mL | 2.4072 mL | 4.8144 mL | 12.0360 mL | |
| 10 mM | 0.2407 mL | 1.2036 mL | 2.4072 mL | 6.0180 mL | |
| 15 mM | 0.1605 mL | 0.8024 mL | 1.6048 mL | 4.0120 mL | |
| 20 mM | 0.1204 mL | 0.6018 mL | 1.2036 mL | 3.0090 mL | |
| 25 mM | 0.0963 mL | 0.4814 mL | 0.9629 mL | 2.4072 mL | |
| 30 mM | 0.0802 mL | 0.4012 mL | 0.8024 mL | 2.0060 mL | |
| 40 mM | 0.0602 mL | 0.3009 mL | 0.6018 mL | 1.5045 mL | |
| 50 mM | 0.0481 mL | 0.2407 mL | 0.4814 mL | 1.2036 mL | |
| 60 mM | 0.0401 mL | 0.2006 mL | 0.4012 mL | 1.0030 mL | |
| 80 mM | 0.0301 mL | 0.1505 mL | 0.3009 mL | 0.7523 mL | |
| 100 mM | 0.0241 mL | 0.1204 mL | 0.2407 mL | 0.6018 mL |