1. GPCR/G Protein
    Neuronal Signaling
    Immunology/Inflammation
  2. Histamine Receptor
  3. Betahistine EP Impurity C

Betahistine EP Impurity C (Synonyms: NSC19005)

Cat. No.: HY-107495
Handling Instructions

Betahistine EP Impurity C (NSC19005) is an impurity of Betahistine. Betahistine is a potent, orally active and well-tolerated histamine H1 receptor agonist and H3 receptor antagonist used for the study of rheumatoid arthritis (RA).

For research use only. We do not sell to patients.

Betahistine EP Impurity C Chemical Structure

Betahistine EP Impurity C Chemical Structure

CAS No. : 5452-87-9

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Description

Betahistine EP Impurity C (NSC19005) is an impurity of Betahistine[1]. Betahistine is a potent, orally active and well-tolerated histamine H1 receptor agonist and H3 receptor antagonist used for the study of rheumatoid arthritis (RA)[2][3].

In Vitro

Betahistine (0-10 μM) inhibits [125I]iodoproxyfan binding to membranes of CHO (rH3(445)R) and CHO (hH3(445)R) cells with IC50 values of 1.9 μM and 3.3 μM, respectively. Lead to Ki values of 1.4 μM and 2.5 μM, respectively[3].

Molecular Weight

241.33

Formula

C₁₅H₁₉N₃

CAS No.

5452-87-9

SMILES

CN(CCC1=CC=CC=N1)CCC2=CC=CC=N2

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

Betahistine EP Impurity CNSC19005NSC 19005NSC-19005Histamine ReceptorimpurityBetahistinehistamineH1H3rheumatoidarthritisRAInhibitorinhibitorinhibit

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