MK 1256

MK 1256 is a highly selective and orally active inhibitor of tissue protease K (Cat K) with an IC50 of 0.62 nM. MK 1256 shows extremely high selectivity towards other tissue proteases (all > 1100 times), with only a slightly lower selectivity for tissue protease F (Cat F) (110 times). MK 1256 exhibits strong anti-bone resorption activity in the osteoporosis model of rhesus monkeys with ovariectomy. MK 1256 can be used for research on osteoporosis.

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  • CAS No.: 919109-76-5
  • Formule: C23H23Cl2F3N4O3S
  • Masse moléculaire:563.42
  • Stockage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

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