CPI-203-PEG1-C3-O-COOH
CPI-203-PEG1-C3-O-COOH is a conjugate of the BRD4 ligand (HY-78695) and the linker (HY-42427). CPI-203-PEG1-C3-O-COOH can be used for synthesizing PROTAC BRD4 degrader ARV-771 (HY-100972).
For research use only. We do not sell to patients.
- CAS No.: 1997304-12-7
- Formula: C26H30ClN5O5S
- Molecular Weight:560.06
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1997304-12-7
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Molecular Weight 560.06
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Formula C26H30ClN5O5S
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SMILES
CC1=C(C)C(C(C2=CC=C(Cl)C=C2)=N[C@@H](CC(NCCOCCCOCC(O)=O)=O)C3=NN=C(C)N34)=C4S1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)