1. Metabolic Enzyme/Protease
  2. Cathepsin
  3. MV061194

MV061194 is a selective cathepsin K inhibitor with a human Ki of 2.5 nM. MV061194 can be used for the research of osteoporosis.

For research use only. We do not sell to patients.

MV061194

MV061194 Chemical Structure

CAS No. : 1021423-50-6

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Description

MV061194 is a selective cathepsin K inhibitor with a human Ki of 2.5 nM. MV061194 can be used for the research of osteoporosis[1].

IC50 & Target[1]

cathepsin K

2.5 nM (Ki)

In Vitro

MV061194 potently and selectively inhibits recombinant human cathepsin K with a Ki of 2.5 nM, showing >4000-fold selectivity over multiple other cathepsin isoforms[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

539.70

Formula

C28H37N5O4S

CAS No.
SMILES

C(N[C@H]1[C@H](CC)OCC1=O)(=O)C2(NC(=O)C3=CC=C(C=C3)C=4N=C(SC4)N5CCN(C)CC5)CCCCC2

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
MV061194
Cat. No.:
HY-15101
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