Naxifylline
Naxifylline (BG9719; CVT-124) is a potent and selective A1-adenosine antagonist with Ki values of 0.67 and 0.45 nM for rat and cloned human A1-receptors, respectively. Naxifylline is a potassium-sparing diuretic for the study of edema associated with congestive heart failure.
For research use only. We do not sell to patients.
- CAS No.: 166374-49-8
- Formula: C18H24N4O3
- Molecular Weight:344.41
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adenosine Receptor Isoforms
More
Biological Activity
|
rat A1 0.67 nM (Ki) |
human A1 0.45 nM (Ki) |
Chemical Information
-
CAS No. 166374-49-8
-
Molecular Weight 344.41
-
Formula C18H24N4O3
-
SMILES
CCCN1C2=C(C(N(C1=O)CCC)=O)NC([C@@H]3[C@@]4([H])[C@@]5([H])[C@]([C@](C3)([H])C4)([H])O5)=N2
-
Synonyms
BG9719; CVT-124
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)