PI3K-IN-9
PI3K-IN-9 (compound 1-14) is a potent and selective PI3Kδ inhibitor with an IC50 of 8.9 nM.
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- No. CAS: 2360875-63-2
- Fòrmula: C19H23N7O
- Peso molecular:365.43
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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PI3Kδ |
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| Sf21 | IC50 |
9 nM
Compound: 29
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Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cells using PIP2 as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr
Inhibition of recombinant human full-length N-terminal GST-tagged p110delta/untagged full-length p85alpha expressed in baculovirus infected Sf21 cells using PIP2 as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr
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[PMID: 31757666] |
Chemical Information
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No. CAS 2360875-63-2
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Peso molecular 365.43
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Fòrmula C19H23N7O
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SMILES
O=C([C@@H]1C[C@H]1C)N(CC2)[C@H](C)CN2C3=CN=C(C#N)C(C4=CN(C)N=C4)=N3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PI3K-IN-9 Related Classifications
HY-133029 Related Classifications
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