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Cat. No.: HY-149421

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BRD7-IN-3

BRD7-IN-3 (compound 1-78) is a dual inhibitor of bromodomain-containing proteins BRD7/BRD9 with IC₅₀s of 1.6 μM and 2.7 μM respectively.

For research use only. We do not sell to patients.

CAS No.: 3032601-04-7
Formula: C₁₈H₁₈N₂O₂
Molecular Weight:294.35

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

BRD7-IN-3 Chemical Structure

CAS No.: 3032601-04-7

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
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Biological Activity

Description

BRD7-IN-3 (compound 1-78) is a dual inhibitor of bromodomain-containing proteins BRD7/BRD9 with IC₅₀s of 1.6 μM and 2.7 μM respectively^[1].

IC₅₀ & Target

IC50: 1.6 μM (BRD7), 2.7 μM (BRD9)^[1]

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Chemical Information

CAS No. 3032601-04-7
Molecular Weight 294.35
Formula C₁₈H₁₈N₂O₂
SMILES

CC1=CC(N(C2=C1C=CC(C3=CC=C(N=C3C)OC)=C2)C)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Ordonez-Rubiano SC, et al. Rational Design and Development of Selective BRD7 Bromodomain Inhibitors and Their Activity in Prostate Cancer. J Med Chem. 2023 Aug 24;66(16):11250-11270.. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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BRD7-IN-3

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Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

BRD7-IN-3 Related Classifications

HY-149421 Related Classifications