4-Methoxywarfarin
4-Methoxywarfarin (compound 15) is a racemic inhibitor of cytochrome P450 2C9 (CYP2C9). 4-Methoxywarfarin inhibits CYP2C9-catalyzed S-warfarin 7-hydroxylation with a Ki of 11 μM. 4-Methoxywarfarin is applicable to studies related to CYP2C9 inhibition, warfarin metabolism, and the structure-activity relationship of CYP2C9 inhibitors.
For research use only. We do not sell to patients.
- CAS No.: 38063-51-3
- Formula: C20H18O4
- Molecular Weight:322.35
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
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- References
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Help & FAQs
Biological Activity
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CYP2C9 11 μM (Ki) |
4-Methoxywarfarin (compound 15) inhibits CYP2C9-catalyzed S-warfarin 7-hydroxylation, with a measured Ki of 11 μM, which is consistent with the Ki of 11 μM predicted by its CoMFA model[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 38063-51-3
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Molecular Weight 322.35
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Formula C20H18O4
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SMILES
O=C1OC2=C(C(OC)=C1C(CC(C)=O)C3=CC=CC=C3)C=CC=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
4-Methoxywarfarin Related Classifications
HY-184843 Related Classifications
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