Opioid Receptor
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Opioid Receptor Inhibitors
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Opioid Receptor Agonists
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Opioid Receptor Antagonists
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Opioid Receptor Ligands
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Opioid Receptor Related Products (367)
Related Products (367)
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Noscapine hydrochloride
0 ImagesNoscapine ((S,R)-Noscapine) hydrochloride is an orally active phthalideisoquinoline alkaloid with potent antitussive. Noscapine hydrochloride exerts its antitussive effects by activating sigma opioid receptors and is a non-competitive Bradykinin inhibitor. Noscapine hydrochloride disrupts microtubule dynamics, induces mitotic arrest and apoptosis. Noscapine hydrochloride possesses anticancer, neuroprotective, anti-inflammatory activities, and can crosse the blood-brain barrier.
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Samidorphan
0 ImagesSynonyms: ALKS-33; RDC-0313Samidorphan (ALKS-33) is an orally active opioid receptor modulator that targets μ-opioid, κ-opioid, and δ-opioid receptors. Samidorphan acts as a μ-opioid receptor antagonist and a partial agonist at κ-opioid and δ-opioid receptors. In vivo, Samidorphan functions primarily as an opioid receptor antagonist and ameliorates depressive behaviors in animals.
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CR 665
0 ImagesSynonyms: JNJ 38488502; FE 200665CR 665 (JNJ 38488502) is a peripherally selective κ-opioid agonist. CR 665 can activate the kappa opioid receptor with EC50 value of 10.9 nM. CR 665 can be used for the research of peripheral pain.
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SCH 221510
0 ImagesSCH 221510 is a potent, orally active and selective NOP (nociceptin opioid receptor) agonist, with an EC50 of 12 nM and Ki of 0.3 nM. SCH 221510 shows an anxiolytic-like effect.
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[Leu5]-Enkephalin, amide
![[Leu5]-Enkephalin, amide](https://file.medchemexpress.com/product_pic/hy-p1470.gif "Click to View [Leu5]-Enkephalin, amide Product Detail")
0 ImagesSynonyms: Leu-Enkephalin amide[Leu5]-Enkephalin, amide is a δ opioid receptor agonist.
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(+)-N-Allylnormetazocine hydrochloride
0 ImagesSynonyms: (+)-SKF 10047 hydrochloride; (+)-N-Allyl-N-normetazocine hydrochloride(+)-N-Allylnormetazocine ((+)-SKF 10047) hydrochloride is a benzomorphan opioid with psychotomi metic effects. (+)-N-Allylnormetazocine hydrochloride is an opioid receptor antagonist with Ki values of 300 nM and 27 μM for σ1 and σ2 opioid receptors, respectively. (+)-N-Allylnormetazocine hydrochloride can be used for the research of neurological disease.
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Anrikefon acetate
0 ImagesSynonyms: HSK21542 acetateAnrikefon (HSK21542) acetate is a kappa opioid receptor agonist with analgesic effect.
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Naloxone hydrochloride (Standard)
0 ImagesNaloxone (hydrochloride) (Standard) is the analytical standard of Naloxone (hydrochloride) (HY-17417). This product is intended for research and analytical applications. Naloxone hydrochloride is an orally active opioid receptor antagonist. Naloxone hydrochloride attenuates spinal cord stimulation‑associated anti‑hyperalgesic effects, antagonizes physiologic effects of endogenous opioid peptides linked to central nervous system injury sequelae, functions as a pressor agent to induce modest elevations in mean arterial blood pressure, exerts neuroprotective effects to improve post‑traumatic neurologic motor function, blocks opioid receptor‑mediated amnesic pathways, enhances memory consolidation, reverses Adrenocorticotropic hormone (ACTH) (HY-106373)‑ and epinephrine‑induced amnesia, and potentiates the memory‑facilitatory effects of ACTH and epinephrine.
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Vanilpyruvic acid
0 ImagesVanilpyruvic acid is a catecholamine metabolite and precursor to vanillactic acid.
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Orphanin FQ(1-11)
0 ImagesOrphanin FQ(1-11), a orphanin FQ or nociceptin (OFQ/N) fragment, is a potent NOP receptor (ORL-1; OP4) agonist, with a Ki of 55 nM. Orphanin FQ(1-11) has no affinity for μ, δ, κ1 and κ3 receptors (Ki>1000 nM). Orphanin FQ(1-11) is analgesic in CD-1 mice.
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ICI-204448
0 ImagesICI-204448 is a κ-opioid agonist with limited access to the CNS, ICI-204448 can displace the binding of the kappa-opioid ligand 3H-bremazocine from guinea pig cerebellum membranes.
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Gluten Exorphin B5
0 ImagesGluten Exorphin B5 is an exogenous opioid peptides derived from wheat gluten, acts on opioid receptor, increases postprandial plasma insulin level in rats.
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GR 89696
0 ImagesGR 89696 is a highly selective κ2 opioid receptor agonist with potential to prevent pruritus.
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Iprindole
0 ImagesIprindole, an opioid receptor agonist, is a tricyclic antidepressant. Iprindole shortens the immobility time in mice forced swimming test, which can be reversed by the opiate antagonist Naloxone (HY-17417A). Iprindole induces lamellar body formation but devoid of lamellar bodies. Iprindole can be used for the research of depression.
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Salvinorin A
0 ImagesSynonyms: Divinorin ASalvinorin A is a potent, unique and short-acting high efficacy kappa-opioid receptor (KOPr) agonist with Ki value of 4.3 nm. Salvinorin A is a non-nitrogenous neoclerodane isolated from Salvia divinorum.
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N-terminally acetylated Leu-enkephalin
0 ImagesSynonyms: Ac-L-Tyr-Gly-Gly-L-Phe-D-Leu-COOHN-terminally acetylated Leu-enkephalin is the N-terminally acetylated form of Leu-enkephalin. Leu-enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.
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LY2940094 tartrate
0 ImagesSynonyms: BTRX-246040 tartrateLY2940094 (BTRX-246040) tartrate is a potent, brain penetrant, selective and orally available N/OFQ peptide (NOP) receptor antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY2940094 tartrate reduces Ethanol self-administration and Ethanol seeking in animal models.
