A-850002
A-850002 is a metabotropic glutamate receptor (mGluR) antagonist (IC50=27 nM) that significantly attenuates spontaneous pain behavior after skin incision in rats. A-850002 can be used for analgesia research.
For research use only. We do not sell to patients.
- CAS No.: 869802-73-3
- Formula: C18H16N4OS
- Molecular Weight:336.41
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Protocols
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
rat mGluR1 41 nM (Ki) |
Chemical Information
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CAS No. 869802-73-3
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Molecular Weight 336.41
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Formula C18H16N4OS
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SMILES
O=C1C2=C(C3=C(C=NC=C3N(C)C)S2)N=CN1C4=CC=C(C)C=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Protocols
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Cell Cytotoxicity Assay
Cytotoxicity assays are usually based on the assessment of cell membrane damage, which can also be indirectly detected by measuring cell viability. Detection methods include MTT assay, CKK-8 assay, LDH assay and ATP assay, etc.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
A-850002 Related Classifications
HY-111256 Related Classifications
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