PF-4522654
PF-4522654 is a potent, selective and brain-permeable 5-HT2C receptor agonist with an EC50 of 16 nM and a Ki of 8 nM. PF-4522654 shows no measurable functional agonism at no 5-HT2A and 5-HT2B receptors. PF-4522654 can be used for the study of stress urinary incontinence (SUI).
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- CAS. Nr.: 1065109-28-5
- Formel: C16H18F2N4
- Molecular Weight:304.34
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Biologische Aktivität
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5-HT2A Receptor |
5-HT2B Receptor |
5-HT2C Receptor |
5-HT2C Receptor 16 nM (EC50) |
5-HT2C Receptor 8 nM (Ki) |
5-HT2B Receptor >10000 nM (EC50) |
Chemical Information
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CAS. Nr. 1065109-28-5
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Molecular Weight 304.34
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Formel C16H18F2N4
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SMILES
FC(C1=NC(CCNCC2)=C2C(NC)=N1)(C3=CC=CC=C3)F
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
PF-4522654 Related Classifications
HY-124947 Related Classifications
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