BET-IN-27
BET-IN-27 (compound 6C) is an oral BET inhibitor with the IC50 values of 3.3 nM (BRD4-BD2)、3.4 nM (BRD4-BD1)、4.1 nM (BRD2-BD1)、20.4 nM (BRD3-BD1) and 42.0 nM (BRDT-BD1), respectively. BET-IN-27 shows anti-proliferative activity.
For research use only. We do not sell to patients.
- CAS No.: 3054869-29-0
- Formula: C21H23N5O3S
- Molecular Weight:425.50
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 3054869-29-0
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Molecular Weight 425.50
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Formula C21H23N5O3S
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SMILES
CN(C(C1=C2C=CN1)=O)C=C2C3=NC4=C(SC(C(C)(C)O)=C4)C(N5CCOCC5)=N3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)