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Cat. No.: HY-184843

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4-Methoxywarfarin

4-Methoxywarfarin (compound 15) is a racemic inhibitor of cytochrome P450 2C9 (CYP2C9). 4-Methoxywarfarin inhibits CYP2C9-catalyzed S-warfarin 7-hydroxylation with a K_i of 11 μM. 4-Methoxywarfarin is applicable to studies related to CYP2C9 inhibition, warfarin metabolism, and the structure-activity relationship of CYP2C9 inhibitors.

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CAS No.: 38063-51-3
Formule: C₂₀H₁₈O₄
Masse moléculaire:322.35

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Please store the product under the recommended conditions in the Certificate of Analysis.

4-Methoxywarfarin Chemical Structure

CAS No.: 38063-51-3

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Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
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- In Vitro
Chemical Information
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Description

IC₅₀ & Target^[1]

CYP2C9

11 μM (Ki)

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In Vitro

4-Methoxywarfarin (compound 15) inhibits CYP2C9-catalyzed S-warfarin 7-hydroxylation, with a measured K_i of 11 μM, which is consistent with the K_i of 11 μM predicted by its CoMFA model^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 38063-51-3
Masse moléculaire 322.35
Formule C₂₀H₁₈O₄
SMILES

O=C1OC2=C(C(OC)=C1C(CC(C)=O)C3=CC=CC=C3)C=CC=C2
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Zhou SF, et al. Substrates, inducers, inhibitors and structure-activity relationships of human cytochrome P450 2C9 and implications in drug development. Current Medicinal Chemistry. 2009;16(27):3480-3675.

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références

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4-Methoxywarfarin

Voir tous les produits spécifiques à Isoform Cytochrome P450