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Cat. No.: HY-127141

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Cizolirtine citrate

(Synonyms: E-4018)

Cizolirtine citrate (E-4018) is an analgesic agent. Cizolirtine citrate has significant analgesic and anti-hyperalgesic action in neuropathic pain models.

For research use only. We do not sell to patients.

CAS No.: 251375-82-3
Formula: C₂₁H₂₉N₃O₈
Molecular Weight:451.47

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (272 KB)

Cizolirtine citrate Chemical Structure

CAS No.: 251375-82-3

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

Description

Cizolirtine citrate (E-4018) is an analgesic agent. Cizolirtine citrate has significant analgesic and anti-hyperalgesic action in neuropathic pain models^[1].

IC₅₀ & Target

5-HT_1B Receptor

All Adenosine Receptor Isoforms :

All 5-HT Receptor Isoforms :

Chemical Information

CAS No. 251375-82-3
Molecular Weight 451.47
Formula C₂₁H₂₉N₃O₈
SMILES

CN1N=CC=C1C(OCCN(C)C)C2=CC=CC=C2.O=C(O)CC(O)(CC(O)=O)C(O)=O
Synonyms

E-4018
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (272 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Shembalkar P, et al. Cizolirtine citrate (E-4018) in the treatment of chronic neuropathic pain. Curr Med Res Opin. 2001;17(4):262-6. [Content Brief]

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Biological Activity
- Description
- IC₅₀ & Target
Chemical Information
Purity & Documentation
References

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Cizolirtine citrate

All Adenosine Receptor Isoforms

All 5-HT Receptor Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

Cizolirtine citrate Related Classifications

HY-127141 Related Classifications