1. Protein Tyrosine Kinase/RTK
  2. FGFR
    VEGFR
  3. FGFR3-IN-2

FGFR3-IN-2 

Cat. No.: HY-147714
Handling Instructions

FGFR3-IN-2 (compound 18b) is a potent and selective FGFR3 inhibitor, with IC50s of 4.1 nM and 570 nM for FGFR3 and VEGFR2, respectively. FGFR3-IN-2 can be used for the research of bladder cancer.

For research use only. We do not sell to patients.

FGFR3-IN-2 Chemical Structure

FGFR3-IN-2 Chemical Structure

CAS No. : 2428742-58-7

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Description

FGFR3-IN-2 (compound 18b) is a potent and selective FGFR3 inhibitor, with IC50s of 4.1 nM and 570 nM for FGFR3 and VEGFR2, respectively. FGFR3-IN-2 can be used for the research of bladder cancer[1].

IC50 & Target[1]

FGFR3

4.1 nM (IC50)

VEGFR2

570 nM (IC50)

Molecular Weight

597.73

Formula

C28H39N9O4S

CAS No.
SMILES

CCNS(=O)(C1=CC=CC=C1NC2=NC(NC3=CC=C(C(OCCN4CCOCC4)=C3)N5CCN(CC5)C)=NC=N2)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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FGFR3-IN-2
Cat. No.:
HY-147714
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