VU0530244
VU0530244 is a potent antagonist of 5-HT2B, with the IC50 of 17.3 nM. VU0530244 is predicted to have very limited potential for brain penetration in human subjects, as is predicted to be substrates for P-gp-mediated efflux in humans.
For research use only. We do not sell to patients.
- CAS No.: 1396886-30-8
- Formula: C22H20FN5O
- Molecular Weight:389.43
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2B Receptor |
5-HT2B Receptor 17.3 nM (IC50) |
Chemical Information
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CAS No. 1396886-30-8
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Molecular Weight 389.43
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Formula C22H20FN5O
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SMILES
O=C(N1CC(C1)C2=NC3=C(N2)C=C(C)C=C3)C4=CC(C5=CC=C(F)C=C5)=NN4C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
VU0530244 Related Classifications
HY-171194 Related Classifications
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