F1324 TFA
F1324 TFA is a potent, high affinity peptidic inhibitor of B cell lymphoma 6 (BCL6), with an IC50 of 1 nM. F1324 TFA exhibits binding t1/2 value of 441 s and has strong inhibition activity against BCL6 PPI.
Para uso exclusivo en investigación. No vendemos a pacientes.
- Fòrmula: C83H121N21O20S.xC2HF3O2
- Peso molecular:1765.04 (free acid)
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
IC50: 1 nM (BCL6)[1]
F1324 TFA binds to BCL6(5-129) with KD and IC50 values of 0.57 nM and 1 nM according to the results of an SPR analysis and cell-free ELISA assay, respectively[1].
F1324 TFA binds BCL6 not only in cell-free but also cellbased conditions[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Peso molecular 1765.04 (free acid)
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Fòrmula C83H121N21O20S.xC2HF3O2
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Sequence Shortening
Ac-LWYTDIRMSWRVP-OH
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)