Pellotine
Pellotine is an alkaloid that can be isolated from Lophophora. Pellotine is the inverse agonist for 5-HT7 receptor with an EC50 of 291 nM. Pellotine exhibits good affinity to 5-HT1DR and 5-HT6R with Ki of 117 nM and 170 nM. Pellotine reduces intracellular cAMP levels, thereby reducing neuronal excitability and neurotransmitter release.
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- No. CAS: 19622-05-0
- Fòrmula: C13H19NO3
- Peso molecular:237.29
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Ver todos los productos específicos de isoformas 5-HT Receptor
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Actividad biológica
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5-HT7 Receptor |
Human 5-HT7 Receptor 291 nM (EC50) |
5-HT1D Receptor 117 nM (Ki) |
5-HT6 Receptor 170 nM (Ki) |
Chemical Information
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No. CAS 19622-05-0
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Peso molecular 237.29
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Fòrmula C13H19NO3
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SMILES
COC1=C(OC)C(O)=C(C(C)N(C)CC2)C2=C1
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pellotine Related Classifications
HY-170908 Related Classifications
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