F1324 TFA
F1324 TFA is a potent, high affinity peptidic inhibitor of B cell lymphoma 6 (BCL6), with an IC50 of 1 nM. F1324 TFA exhibits binding t1/2 value of 441 s and has strong inhibition activity against BCL6 PPI.
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- 分子式: C83H121N21O20S.xC2HF3O2
- 分子量:1765.04 (free acid)
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
IC50: 1 nM (BCL6)[1]
F1324 TFA binds to BCL6(5-129) with KD and IC50 values of 0.57 nM and 1 nM according to the results of an SPR analysis and cell-free ELISA assay, respectively[1].
F1324 TFA binds BCL6 not only in cell-free but also cellbased conditions[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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分子量 1765.04 (free acid)
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分子式 C83H121N21O20S.xC2HF3O2
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シーケンスの短縮
Ac-LWYTDIRMSWRVP-OH
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)