LUF8100
Based on 1 Customer Validation
LUF8100 is a dual-target antagonist of CCR2/CCR5 with pKi values for CCR2 and CCR5 of 5.23 and 4.97 respectively. LUF8100 can be used for research on immune homeostasis and cancer.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 98.64%
- CAS 番号: 2954281-30-0
- 分子式: C18H18ClF3N2O2S
- 分子量:418.86
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
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GPCR/G Protein Compound Library
HY-L006
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Immunology/Inflammation Compound Library
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Anti-Cancer Compound Library
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Small Molecule Immuno-Oncology Compound Library
HY-L031
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Anti-Pulmonary Fibrosis Compound Library
HY-L125
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Chemokine Compound Library
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Membrane Protein-targeted Compound Library
HY-L149
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Membrane Receptor-targeted Compound Library
HY-L150
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Cytokine Inhibitors Library
HY-L161
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Multi-Target Compound Library
HY-L176
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Bioactive Compound Library Max
HY-L181
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MCE Bioactive Compound Library
HY-L001V
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Bioactive Compound Library
HY-L001
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Non-Alcoholic Fatty Liver Disease (NAFLD) Compound Library
HY-L199
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High-Throughput Bioactive Compound Library
HY-L205
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Anti-Rheumatic Arthritis Compound Library
HY-L210
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Lactylation Compound Library
HY-L249
生物活性
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CCR2 5.23 (pKi) |
CCR5 4.97 (pKi) |
化学情報
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CAS 番号 2954281-30-0
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性状 Solid
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分子量 418.86
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分子式 C18H18ClF3N2O2S
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Color Off-white to pink
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SMILES
O=S(NC1=CC(N2CCCCC2)=CC=C1)(C3=CC=C(Cl)C(C(F)(F)F)=C3)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : ≥ 100 mg/mL (238.74 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
* "≥" means soluble, but saturation unknown.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (271 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.3874 mL | 11.9372 mL | 23.8743 mL | 59.6858 mL |
| 5 mM | 0.4775 mL | 2.3874 mL | 4.7749 mL | 11.9372 mL | |
| 10 mM | 0.2387 mL | 1.1937 mL | 2.3874 mL | 5.9686 mL | |
| 15 mM | 0.1592 mL | 0.7958 mL | 1.5916 mL | 3.9791 mL | |
| 20 mM | 0.1194 mL | 0.5969 mL | 1.1937 mL | 2.9843 mL | |
| 25 mM | 0.0955 mL | 0.4775 mL | 0.9550 mL | 2.3874 mL | |
| 30 mM | 0.0796 mL | 0.3979 mL | 0.7958 mL | 1.9895 mL | |
| 40 mM | 0.0597 mL | 0.2984 mL | 0.5969 mL | 1.4921 mL | |
| 50 mM | 0.0477 mL | 0.2387 mL | 0.4775 mL | 1.1937 mL | |
| 60 mM | 0.0398 mL | 0.1990 mL | 0.3979 mL | 0.9948 mL | |
| 80 mM | 0.0298 mL | 0.1492 mL | 0.2984 mL | 0.7461 mL | |
| 100 mM | 0.0239 mL | 0.1194 mL | 0.2387 mL | 0.5969 mL |
LUF8100 関連分類
HY-179607 関連分類
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