LY320954
LY320954 is a selective 5-HT2A receptor antagonist, with a Ki of 96 nM. LY320954 potently inhibits Ca2+ influx in the functional assay (EC50 of 35.5 nM). LY320954 inhibits 5-HT-induced paw swelling in rats, with ED50 of 4.8 mg/kg.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 182633-59-6
- Formel: C21H26N4O3
- Molecular Weight:382.46
-
Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Alle 5-HT Receptor Isoform-spezifische Produkte anzeigen
More
Biologische Aktivität
|
5-HT2A Receptor |
5-HT2A Receptor 96 nM (Ki) |
5-HT2B Receptor 1642 nM (Ki) |
5-HT2C Receptor 257 nM (Ki) |
Chemical Information
-
CAS. Nr. 182633-59-6
-
Molecular Weight 382.46
-
Formel C21H26N4O3
-
SMILES
CCCC1=C(O)C(C(CC)=O)=CC=C1COC2=CC=C(/C=N/NC(N)=N)C=C2
-
Versand
Room temperature in continental US; may vary elsewhere.
-
Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)