LY320954
LY320954 is a selective 5-HT2A receptor antagonist, with a Ki of 96 nM. LY320954 potently inhibits Ca2+ influx in the functional assay (EC50 of 35.5 nM). LY320954 inhibits 5-HT-induced paw swelling in rats, with ED50 of 4.8 mg/kg.
For research use only. We do not sell to patients.
- CAS No.: 182633-59-6
- Formula: C21H26N4O3
- Molecular Weight:382.46
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT2A Receptor |
5-HT2A Receptor 96 nM (Ki) |
5-HT2B Receptor 1642 nM (Ki) |
5-HT2C Receptor 257 nM (Ki) |
Chemical Information
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CAS No. 182633-59-6
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Molecular Weight 382.46
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Formula C21H26N4O3
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SMILES
CCCC1=C(O)C(C(CC)=O)=CC=C1COC2=CC=C(/C=N/NC(N)=N)C=C2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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