1 Result for "

Relative Cellular Potencies

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Relative Cellular Potencies" in MCE Product Catalog:

Cat. No.: HY-103453
CAS No.: 524047-78-7
Target:  

Estrogen Receptor/ERR

Research Areas:  

Endocrinology

(R)-DPN (compound 3) is a selective ERβ ligand with EC50s of 2.9, 0.8 nM for ERα and ERβ, respectively. (R)-DPN shows a very high affinity and potency preference for ERβ over ERα. (R)-DPN shows cytoxicity for HEC-1 and U2OS cells with EC50s of 286, 205 nM, respectively .
loading...
    loading...