1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor

Tianeptine sodium salt 

Cat. No.: HY-90003A Purity: 99.88%
Handling Instructions

Tianeptine sodium salt is a selective facilitator of 5-HT uptake in vitro and in vivo.

For research use only. We do not sell to patients.

Tianeptine sodium salt Chemical Structure

Tianeptine sodium salt Chemical Structure

CAS No. : 30123-17-2

Size Stock
10 mM * 1 mL in DMSO Get quote
10 mg USD 60 Get quote
50 mg USD 78 Get quote
100 mg USD 114 Get quote

* Please select Quantity before adding items.

Other Forms of Tianeptine sodium salt:

Customer Validation

    Tianeptine sodium salt purchased from MCE. Usage Cited in: bioRxiv. April 7, 2018.

    Antidepressant Tianeptine rescues the reduced BDNF protein level and intracellular transport in different complementary HD models.
    • Biological Activity

    • Technical Information

    • Purity & Documentation

    • References

    Description

    Tianeptine sodium salt is a selective facilitator of 5-HT uptake in vitro and in vivo. IC50 Value: Target: 5-HT Receptor Tianeptine has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM) and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo.

    Clinical Trial
    Solvent & Solubility
    In Vitro: 

    H2O : ≥ 235 mg/mL (512.06 mM)

    *"≥" means soluble, but saturation unknown.

    Preparing
    Stock Solutions
    Concentration Solvent Mass 1 mg 5 mg 10 mg
    1 mM 2.1790 mL 10.8949 mL 21.7898 mL
    5 mM 0.4358 mL 2.1790 mL 4.3580 mL
    10 mM 0.2179 mL 1.0895 mL 2.1790 mL
    *Please refer to the solubility information to select the appropriate solvent.
    References
    Molecular Weight

    458.93

    Formula

    C₂₁H₂₄ClN₂NaO₄S

    CAS No.

    30123-17-2

    SMILES

    O=C(CCCCCCNC(C1=CC=CC=C1N2C)C3=CC=C(C=C3S2(=O)=O)Cl)[O-].[Na+]

    Storage
    Powder -20°C 3 years
      4°C 2 years
    In solvent -80°C 6 months
      -20°C 1 month
    Shipping

    Room temperature in continental US; may vary elsewhere

    • Molarity Calculator

    • Dilution Calculator

    The molarity calculator equation

    Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

    Mass   Concentration   Volume   Molecular Weight *
    = × ×

    The dilution calculator equation

    Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

    This equation is commonly abbreviated as: C1V1 = C2V2

    Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
    × = ×
    C1   V1   C2   V2

    Inquiry Online

    Your information is safe with us. * Required Fields.

    Product name

     

    Salutation

    Applicant name *

     

    Email address *

    Phone number *

     

    Organization name *

    Country or Region *

     

    Requested quantity *

    Remarks

    Bulk Inquiry

    Inquiry Information

    Product Name:
    Tianeptine sodium salt
    Cat. No.:
    HY-90003A
    Quantity:

    Tianeptine sodium salt

    Cat. No.: HY-90003A