1. GPCR/G Protein
    Neuronal Signaling
  2. 5-HT Receptor
  3. Tianeptine sodium salt

Tianeptine sodium salt 

Cat. No.: HY-90003A Purity: 99.82%
Handling Instructions

Tianeptine sodium salt is a selective facilitator of 5-HT uptake in vitro and in vivo.

For research use only. We do not sell to patients.

Tianeptine sodium salt Chemical Structure

Tianeptine sodium salt Chemical Structure

CAS No. : 30123-17-2

Size Stock
10 mM * 1  mL in DMSO Get quote
10 mg USD 60 Get quote
50 mg USD 78 Get quote
100 mg USD 114 Get quote

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Other Forms of Tianeptine sodium salt:

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Description

Tianeptine sodium salt is a selective facilitator of 5-HT uptake in vitro and in vivo. IC50 Value: Target: 5-HT Receptor Tianeptine has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM) and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo.

IC50 & Target

serotonin

 

Clinical Trial
Molecular Weight

458.93

Formula

C₂₁H₂₄ClN₂NaO₄S

CAS No.

30123-17-2

SMILES

O=C(CCCCCCNC(C1=CC=CC=C1N2C)C3=CC=C(C=C3S2(=O)=O)Cl)O[Na]

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (217.90 mM; Need ultrasonic)

H2O : 100 mg/mL (217.90 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1790 mL 10.8949 mL 21.7898 mL
5 mM 0.4358 mL 2.1790 mL 4.3580 mL
10 mM 0.2179 mL 1.0895 mL 2.1790 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (5.45 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (5.45 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (5.45 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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  • Molarity Calculator

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Tianeptine5-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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Tianeptine sodium salt
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HY-90003A
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