Tiropramide hydrochloride
Based on 1 Customer Validation
Tiropramide (CR 605) hydrochloride is a tyrosine derivative with antispastic properties. Tiropramide hydrochloride inhibits phosphodiesterase activity involved in cAMP catabolism in rabbit colon homogenates. Tiropramide hydrochloride relaxes smooth muscle in rabbit isolated colon. Tiropramide hydrochloride can be used for the research of irritable colon and biliary dyskinesia.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 53567-47-8
- 分子式: C28H42ClN3O3
- 分子量:504.10
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保管条件:
4°C, sealed storage, away from moisture and light
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
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溶剤 & 溶解度
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
製品説明
体外実験
Tiropramide hydrochloride inhibits phosphodiesterase activity in rabbit colon homogenates and increases ATP- and Mg2+-dependent calcium binding to rabbit colon sarcoplasmic reticulum microsomal fractions[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 53567-47-8
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性状 Solid
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分子量 504.10
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分子式 C28H42ClN3O3
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SMILES
O=C(C1=CC=CC=C1)NC(CC2=CC=C(C=C2)OCCN(CC)CC)C(N(CCC)CCC)=O.Cl
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別名
CR 605 hydrochloride
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
4°C, sealed storage, away from moisture and light
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)
溶剤 & 溶解度
体外:
DMSO : 125 mg/mL (247.97 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (269 KB)
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SDS (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.9837 mL | 9.9187 mL | 19.8373 mL | 49.5933 mL |
| 5 mM | 0.3967 mL | 1.9837 mL | 3.9675 mL | 9.9187 mL | |
| 10 mM | 0.1984 mL | 0.9919 mL | 1.9837 mL | 4.9593 mL | |
| 15 mM | 0.1322 mL | 0.6612 mL | 1.3225 mL | 3.3062 mL | |
| 20 mM | 0.0992 mL | 0.4959 mL | 0.9919 mL | 2.4797 mL | |
| 25 mM | 0.0793 mL | 0.3967 mL | 0.7935 mL | 1.9837 mL | |
| 30 mM | 0.0661 mL | 0.3306 mL | 0.6612 mL | 1.6531 mL | |
| 40 mM | 0.0496 mL | 0.2480 mL | 0.4959 mL | 1.2398 mL | |
| 50 mM | 0.0397 mL | 0.1984 mL | 0.3967 mL | 0.9919 mL | |
| 60 mM | 0.0331 mL | 0.1653 mL | 0.3306 mL | 0.8266 mL | |
| 80 mM | 0.0248 mL | 0.1240 mL | 0.2480 mL | 0.6199 mL | |
| 100 mM | 0.0198 mL | 0.0992 mL | 0.1984 mL | 0.4959 mL |
Tiropramide hydrochloride 関連分類
HY-43934 関連分類
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