country

Change Language

EN - English
FR - Français
DE - Deutsch
ES - Español
JA - 日本語
KO - 한국어

Country or Region:

United States

Product Name	Size / Unit Price	Qty

Total: USD 0.00 Checkout

Art. -Nr.: HY-116780

Copy Link Print Information

Prothipendyl

Prothipendyl is a tricyclic azaphenothiazine neuroleptic agent. Prothipendyl is a substrate of the CYP isozymes CYP1A2, CYP2D6, CYP2C19 and CYP3A4. Prothipendyl has sedating and psychomotorically damping effects. Prothipendyl can be used for psychomotoric agitation, sleep disorder and anxiety research .

Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.

CAS. Nr.: 303-69-5
Formel: C₁₆H₁₉N₃S
Molecular Weight:285.41

Speicherung:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

Prothipendyl Chemical Structure

CAS. Nr.: 303-69-5

Größe

Preis

Verfügbarkeit

Menge

Amount: USD 0.00

* Bitte wählen Sie Menge, bevor Sie Artikel hinzufügen.

Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biologische Aktivität
- Beschreibung
- Cellular Effect
- Clinical Trial
Chemical Information
Reinheit & Dokumentation
Verweise
Calculators
Help & FAQs
Classifications
Bioz

Biologische Aktivität

Beschreibung

Alle Cytochrome P450 Isoform-spezifische Produkte anzeigen :

Cellular Effect

Cell Line	Type	Value	Description	References
C32	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human C32 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human C32 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
HFF-1	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human HFF1 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human HFF1 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
MCF7	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human MCF7 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human MCF7 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
SNB-19	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human SNB19 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human SNB19 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
T47D	IC₅₀	32.3 μg/mL Compound: Prothipendyl	Cytotoxicity against human T47D cells Cytotoxicity against human T47D cells	[PMID: 28734245]

Clinical Trial

NCT Number	Sponsor	Condition	Start Date	Phase A549
NCT01329991	Plexxikon\|		2011-05	PHASE1

Chemical Information

CAS. Nr. 303-69-5
Molecular Weight 285.41
Formel C₁₆H₁₉N₃S
SMILES

CN(C)CCCN1C2=NC=CC=C2SC3=CC=CC=C13
Versand

Room temperature in continental US; may vary elsewhere.
Speicherung

Please store the product under the recommended conditions in the Certificate of Analysis.

Reinheit & Dokumentation

Select Batch:

Reinheit: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (267 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

Verweise

[1]. Krämer M, et al. Range of therapeutic prothipendyl and prothipendyl sulfoxide concentrations in clinical blood samples. Drug Test Anal. 2018 Jun;10(6):1009-1016. [Content Brief]

Calculators

Molaritätsrechner

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Konzentration Konzentration

Volumen Volumen

Molecular Weight Molecular Weight

Verdünnungsrechner

Konzentration _{(Stammlösung)} × Volumen _{(Stammlösung)} = Konzentration _{(Ziellösung)} × Volumen _{(Ziellösung)}

Konzentration _{(Stammlösung)} Konzentration _{(Stammlösung)}

Volumen _{(Stammlösung)} Volumen _{(Stammlösung)}

Konzentration _{(Ziellösung)} Konzentration _{(Ziellösung)}

Volumen _{(Ziellösung)} Volumen _{(Ziellösung)}

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

MOQ

Minimum order quantity

100 mg

Angebot einholen Auf Lager

Other size

Angebot einholen

Amount: USD 0.00

Biologische Aktivität
- Beschreibung
- Clinical Trial
Chemical Information
Reinheit & Dokumentation
Verweise

Produktname:
Art. -Nr.:
Menge:
MCE Japan Authorized Agent:

Produktname:
CAS. Nr.:
Species:
Reinheit:
Menge:

Prothipendyl

Alle Cytochrome P450 Isoform-spezifische Produkte anzeigen

Biologische Aktivität

Chemical Information

Reinheit & Dokumentation

Verweise

Calculators

Help & FAQs

Prothipendyl Related Classifications

HY-116780 Related Classifications