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  3. BRD4-BD1-IN-2

BRD4-BD1-IN-2 

Cat. No.: HY-143300
Handling Instructions

BRD4-BD1-IN-2 is a selective BRD4-BD1 inhibitor, with an IC50 of 2.51 µM (20-times greater than that of BD2). BRD4-BD1-IN-2 can be used in studies of cancer and cardiovascular diseases.

For research use only. We do not sell to patients.

BRD4-BD1-IN-2 Chemical Structure

BRD4-BD1-IN-2 Chemical Structure

CAS No. : 2761321-26-8

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Description

BRD4-BD1-IN-2 is a selective BRD4-BD1 inhibitor, with an IC50 of 2.51 µM (20-times greater than that of BD2). BRD4-BD1-IN-2 can be used in studies of cancer and cardiovascular diseases[1].

IC50 & Target

BRD4-BD1

2.51 μM (IC50)

BRD4-BD2

>50 μM (IC50)

Molecular Weight

583.07

Formula

C20H15Br3N4O2

CAS No.
SMILES

CN1C(N(C(C2=C1N=C(N2CC3=CC=C(C=C3)Br)Br)=O)CC4=CC=C(C=C4)Br)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Product Name:
BRD4-BD1-IN-2
Cat. No.:
HY-143300
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