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Cat. No.: HY-182371

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BRD4 ligand 15

BRD4 ligand 15 (compound 5) is a BRD4 ligand and alkyne-modified chalcone derivative, which serves as a building block for the synthesis of BRD4-targeting PROTAC TKP-5 (HY-182370).

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CAS No.: 3076613-24-3
Formule: C₂₅H₂₇NO₅
Masse moléculaire:421.49

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Please store the product under the recommended conditions in the Certificate of Analysis.

BRD4 ligand 15 Chemical Structure

CAS No.: 3076613-24-3

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Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
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Activité biologique

Description

BRD4 ligand 15 (compound 5) is a BRD4 ligand and alkyne-modified chalcone derivative, which serves as a building block for the synthesis of BRD4-targeting PROTAC TKP-5 (HY-182370)^[1].

IC₅₀ & Target^[1]

BRD4

BRD2

BRD3

BRDT

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Chemical Information

CAS No. 3076613-24-3
Masse moléculaire 421.49
Formule C₂₅H₂₇NO₅
SMILES

O=C(C)NCCC1=C(C(/C=C/C2=CC=C(OCC#C)C=C2)=O)C=C(OCC)C(OC)=C1
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Yamakoshi H, et al. Alkyne Two-Phase Strategy: Rapid Generation of TK-285-Derived PROTACs as BRD4 Degraders. J Med Chem. Published online March 19, 2026. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Volume Volume

Molecular Weight Molecular Weight

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Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Activité biologique
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- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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BRD4 ligand 15

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