Pellotine
Pellotine is an alkaloid that can be isolated from Lophophora. Pellotine is the inverse agonist for 5-HT7 receptor with an EC50 of 291 nM. Pellotine exhibits good affinity to 5-HT1DR and 5-HT6R with Ki of 117 nM and 170 nM. Pellotine reduces intracellular cAMP levels, thereby reducing neuronal excitability and neurotransmitter release.
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- CAS No.: 19622-05-0
- Formule: C13H19NO3
- Masse moléculaire:237.29
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Stockage:
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Activité biologique
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Chemical Information
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Activité biologique
Description
IC50 & Target
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5-HT7 Receptor |
Human 5-HT7 Receptor 291 nM (EC50) |
5-HT1D Receptor 117 nM (Ki) |
5-HT6 Receptor 170 nM (Ki) |
Chemical Information
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CAS No. 19622-05-0
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Masse moléculaire 237.29
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Formule C13H19NO3
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SMILES
COC1=C(OC)C(O)=C(C(C)N(C)CC2)C2=C1
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pellotine Related Classifications
HY-170908 Related Classifications
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