VU0463841
VU0463841 is a potent, selective and brain-penetrant mGlu5 negative allosteric modulator (NAM) with an IC50 of 13 nM. VU0463841 is ineffective against mGlu1-4 and mGlu7-8. VU0463841 has the potential for the Cocaine addiction research.
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- CAS. Nr.: 1439095-16-5
- Formel: C13H8ClFN4O
- Molecular Weight:290.68
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biologische Aktivität
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mGlu5 Receptor 13 nM (IC50) |
Chemical Information
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CAS. Nr. 1439095-16-5
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Molecular Weight 290.68
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Formel C13H8ClFN4O
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SMILES
O=C(NC1=NC=C(C=C1)Cl)NC2=CC(F)=CC(C#N)=C2
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)