Pellotine
Pellotine is an alkaloid that can be isolated from Lophophora. Pellotine is the inverse agonist for 5-HT7 receptor with an EC50 of 291 nM. Pellotine exhibits good affinity to 5-HT1DR and 5-HT6R with Ki of 117 nM and 170 nM. Pellotine reduces intracellular cAMP levels, thereby reducing neuronal excitability and neurotransmitter release.
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- CAS. Nr.: 19622-05-0
- Formel: C13H19NO3
- Molecular Weight:237.29
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Biologische Aktivität
Beschreibung
IC50 & Target
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5-HT7 Receptor |
Human 5-HT7 Receptor 291 nM (EC50) |
5-HT1D Receptor 117 nM (Ki) |
5-HT6 Receptor 170 nM (Ki) |
Chemical Information
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CAS. Nr. 19622-05-0
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Molecular Weight 237.29
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Formel C13H19NO3
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SMILES
COC1=C(OC)C(O)=C(C(C)N(C)CC2)C2=C1
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
Pellotine Related Classifications
HY-170908 Related Classifications
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