CAY10590
Based on 1 Customer Validation
CAY10590 (GK115) is an inhibitor of secreted phospholipase A2 (sPLA2) and can be used for the research of chronic inflammatory kidney diseases.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 98.0%
- CAS 番号: 1101136-50-8
- 分子式: C21H33NO3
- 分子量:347.49
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保管条件:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
Phospholipase アイソフォーム固有の製品をすべて表示
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生物活性
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sPLA2 |
CAY10590 (GK115) (0-10 μM; 24 h) inhibits IL-1β/forskolin-stimulated PGE2 formation in mesangial cells[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 1101136-50-8
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性状 Solid
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分子量 347.49
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分子式 C21H33NO3
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Color White to off-white
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SMILES
CCCC[C@@H](NC(CCCCCCC1=CC=CC=C1)=O)CCC(O)=O
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別名
GK115
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 20 mg/mL (57.56 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (267 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.8778 mL | 14.3889 mL | 28.7778 mL | 71.9445 mL |
| 5 mM | 0.5756 mL | 2.8778 mL | 5.7556 mL | 14.3889 mL | |
| 10 mM | 0.2878 mL | 1.4389 mL | 2.8778 mL | 7.1945 mL | |
| 15 mM | 0.1919 mL | 0.9593 mL | 1.9185 mL | 4.7963 mL | |
| 20 mM | 0.1439 mL | 0.7194 mL | 1.4389 mL | 3.5972 mL | |
| 25 mM | 0.1151 mL | 0.5756 mL | 1.1511 mL | 2.8778 mL | |
| 30 mM | 0.0959 mL | 0.4796 mL | 0.9593 mL | 2.3982 mL | |
| 40 mM | 0.0719 mL | 0.3597 mL | 0.7194 mL | 1.7986 mL | |
| 50 mM | 0.0576 mL | 0.2878 mL | 0.5756 mL | 1.4389 mL |