Deltasonamide 2
Based on 1 publication(s) in Google Scholar
Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.
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- CAS 番号: 2088485-34-9
- 分子式: C30H39ClN6O4S2
- 分子量:647.25
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
MedChemExpress（MCE）の使用を引用している文献 Deltasonamide 2
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生物活性
Kd: ~385 pM (PDEδ)[1]
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| AGS | IC50 |
1.2 μM
Compound: Deltasonamide 2
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Antiproliferative activity against human AGS cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human AGS cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
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[PMID: 34965125] |
| MIA PaCa-2 | IC50 |
507 nM
Compound: Deltasonamide 2
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Antiproliferative activity against human MIA PaCa-2 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human MIA PaCa-2 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
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[PMID: 34965125] |
| NCI-H358 | IC50 |
954 nM
Compound: Deltasonamide 2
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Antiproliferative activity against human NCI-H358 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human NCI-H358 cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
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[PMID: 34965125] |
| PaTu 8988t | IC50 |
1.2 μM
Compound: Deltasonamide 2
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Antiproliferative activity against human PaTu 8988t cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
Antiproliferative activity against human PaTu 8988t cells assessed as reduction in cell viability measured after 3 days by Celltiter-Glo assay
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[PMID: 34965125] |
化学情報
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CAS 番号 2088485-34-9
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性状 Solid
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分子量 647.25
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分子式 C30H39ClN6O4S2
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Color White to off-white
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SMILES
O=S(C1=CC=C(S(=O)(N(CC2=CC=C(Cl)C=C2)C3CCCC3)=O)C=C1)(N([C@H]4CC[C@H](N)CC4)CC5=NC(NC)=NC=C5)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (1)
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Journal Impact Factor
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Most Recent
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J Med Chem
2022 Jan 13;65(1):747-756. PMID: 34965125
純度とドキュメンテーション
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データシート (267 KB)
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SDS (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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取扱説明書 (2659 KB)
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
Deltasonamide 2 関連分類
HY-122641A 関連分類
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