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製品番号: HY-116780

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Prothipendyl

Prothipendyl is a tricyclic azaphenothiazine neuroleptic agent. Prothipendyl is a substrate of the CYP isozymes CYP1A2, CYP2D6, CYP2C19 and CYP3A4. Prothipendyl has sedating and psychomotorically damping effects. Prothipendyl can be used for psychomotoric agitation, sleep disorder and anxiety research .

商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。

CAS 番号: 303-69-5
分子式: C₁₆H₁₉N₃S
分子量:285.41

保管条件:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (267 KB)

Prothipendyl 構造式

CAS 番号: 303-69-5

容量

価格（税別）

在庫状況

数量

Amount: USD 0.00

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

生物活性

製品説明

Cytochrome P450 アイソフォーム固有の製品をすべて表示 :

Cellular Effect

Cell Line	Type	Value	Description	References
C32	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human C32 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human C32 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
HFF-1	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human HFF1 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human HFF1 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
MCF7	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human MCF7 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human MCF7 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
SNB-19	IC₅₀	>=23 μg/mL Compound: Prothipendyl	Cytotoxicity against human SNB19 cells incubated for 72 hrs by WST1 dye based assay Cytotoxicity against human SNB19 cells incubated for 72 hrs by WST1 dye based assay	[PMID: 28734245]
T47D	IC₅₀	32.3 μg/mL Compound: Prothipendyl	Cytotoxicity against human T47D cells Cytotoxicity against human T47D cells	[PMID: 28734245]

臨床実験

NCT Number	Sponsor	Condition	Start Date	Phase A549
NCT01329991	Plexxikon\|		2011-05	PHASE1

化学情報

CAS 番号 303-69-5
分子量 285.41
分子式 C₁₆H₁₉N₃S
SMILES

CN(C)CCCN1C2=NC=CC=C2SC3=CC=CC=C13
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.

純度とドキュメンテーション

バッチを選択:

純度: 99.98%

Assay: 99.98%

ee.: 99.98%

データシート (267 KB)
COA (2659 KB)
元素分析報告書 (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
取扱説明書 (2659 KB)

参考文献

[1]. Krämer M, et al. Range of therapeutic prothipendyl and prothipendyl sulfoxide concentrations in clinical blood samples. Drug Test Anal. 2018 Jun;10(6):1009-1016. [Content Brief]

Calculators

モル濃度計算機

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

濃度濃度

体積体積

分子量分子量

希釈計算機

濃度 _(開始) × 体積 _(開始) = 濃度 _(終了) × 体積 _(終了)

濃度 _(開始) 濃度 _(開始)

体積 _(開始) 体積 _(開始)

濃度 _(終了) 濃度 _(終了)

体積 _(終了) 体積 _(終了)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

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100 mg

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生物活性
- 製品説明
- 臨床実験
化学情報
純度とドキュメンテーション
参考文献

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Prothipendyl

Cytochrome P450 アイソフォーム固有の製品をすべて表示

生物活性

化学情報

純度とドキュメンテーション

参考文献

Calculators

Help & FAQs

Prothipendyl 関連分類

HY-116780 関連分類