2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation Anti-infection Others
  3. Dopamine Receptor Histamine Receptor Bacterial Amyloid-β Drug Derivative
  4. Norzine dimalate

Norzine dimalate  (Synonyms: Thiethylperazine dimalate)

Cat. No.: HY-A0188
Handling Instructions Technical Support

Norzine dimalate (Thiethylperazine dimalate), a Phenothiazine (HY-Y0055) derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Norzine dimalate is also a selective ABCC1activator that reduces amyloid-β load in mice. Norzine dimalate has anti-emetic, antipsychotic and antimicrobial effects.

For research use only. We do not sell to patients.

Norzine dimalate

Norzine dimalate Chemical Structure

CAS No. : 52239-63-1

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Norzine dimalate Related Antibodies

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Dopamine Receptor D1 Receptor D2 Receptor D3 Receptor D4 Receptor D5 Receptor

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H1 Receptor H2 Receptor H3 Receptor H4 Receptor Histamine Receptor

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Description

Norzine dimalate (Thiethylperazine dimalate), a Phenothiazine (HY-Y0055) derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Norzine dimalate is also a selective ABCC1activator that reduces amyloid-β load in mice. Norzine dimalate has anti-emetic, antipsychotic and antimicrobial effects[1][2][3].

IC50 & Target[1][2][3]

H1 Receptor

 

D2 Receptor

 

Clinical Trial
Molecular Weight

667.79

Formula

C30H41N3O10S2
CAS No.
SMILES

O=C(O)C(O)CC(O)=O.CN1CCN(CCCN2C3=C(C=CC=C3)SC4=CC=C(SCC)C=C24)CC1.O=C(O)C(O)CC(O)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Norzine dimalate Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Norzine dimalate52239-63-1Thiethylperazine dimalateDopamine ReceptorHistamine ReceptorBacterialAmyloid-βDrug Derivativeβ-amyloid peptideAβAbetaDrug derivativeAnti-emeticphenothiazineD2-receptorH1-receptorpregnancycleftAlzheimerdiseaseAβ42ABCC1antipsychoticInhibitorinhibitorinhibit

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