Pimavanserin-d4
Pimavanserin-d4 (ACP-103-d4) is the deuterium labeled Pimavanserin (HY-14557). Pimavanserin is a selective, brain-penetrant, inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively.
For research use only. We do not sell to patients.
- Formula: C25H30D4FN3O2
- Molecular Weight:431.58
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
1. This compound can be used as a tracer
2. This compound can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
Chemical Information
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Unlabeled Cas 706779-91-1
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Molecular Weight 431.58
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Formula C25H30D4FN3O2
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SMILES
CC(C)COC1=CC=C(CNC(N(CC2=C([2H])C([2H])=C(F)C([2H])=C2[2H])C3CCN(C)CC3)=O)C=C1
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Synonyms
ACP-103-d4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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