RS-64459-193
RS-64459-193 is a 5-HT1A receptor partial agonist with a Ki of 24.9 nM. RS-64459-193 also shows high affinity for 5-HT2C, 5-HT2A and 5-HT7 with pKi values of 6.87, 7.02, and 7.18, respectively. RS-64459-193 is almost devoid of activity at the m 5-HT3 receptor.
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- CAS. Nr.: 123882-89-3
- Formel: C26H36Cl2N2O2
- Molecular Weight:479.48
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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Chemical Information
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Help & FAQs
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Biologische Aktivität
Beschreibung
IC50 & Target
[1]|
5-HT1A Receptor |
5-HT2A Receptor |
5-HT2C Receptor |
5-HT7 Receptor |
5-HT1A Receptor 24.9 nM (Ki, CHO cells) |
human 5-HT1A Receptor 7.6 (pKi, Sf9) |
human 5-HT1A Receptor 7.04 (pKi) |
5-HT2C Receptor 6.87 (pKi) |
Rat 5-HT2A 7.02 (pKi) |
Human 5-HT7 Receptor 7.18 (pKi) |
5-HT3 Receptor <4 (pKi) |
Chemical Information
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CAS. Nr. 123882-89-3
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Molecular Weight 479.48
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Formel C26H36Cl2N2O2
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SMILES
O=C1N(C(CC2(CCCC2)C1)=O)CCCCN3CC4C5=C(CCC4)C=CC(Cl)=C5CC3.[H]Cl
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)
RS-64459-193 Related Classifications
HY-120498 Related Classifications
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