(S)-GSK1379725A
(S)-GSK1379725A (compound AU1) is a selective bromodomain and PHD finger containing transcription factor (BPTF) bromodomain inhibitor with a Kd of 2.8 μM. (S)-GSK1379725A shows to be selective for BPTF over BRD4 bromodomain. (S)-GSK1379725A shows antimalarial activity.
For research use only. We do not sell to patients.
- CAS No.: 2359618-49-6
- Formula: C23H23FN6O3
- Molecular Weight:450.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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Plasmodium |
Chemical Information
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CAS No. 2359618-49-6
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Molecular Weight 450.47
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Formula C23H23FN6O3
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SMILES
COC(C1=CC=CC(NC(N[C@@H](CC2)CN2C3=NC(NC4=CC=C(C=C4)F)=NC=C3)=O)=C1)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)