SB-272183
SB-272183 is a selective 5-HT1A, 5-HT1B and 5-HT1D receptor antagonist. In addition, SB-272183 is also a potent and selective ligand for 5-HT1A, 5-HT1B and 5-HT1D receptors in human recombinant and native tissues with pKi values of 8.0, 8.1 and 8.7, respectively. SB-272183 can be used in antidepressant research.
For research use only. We do not sell to patients.
- CAS No.: 216058-27-4
- Formula: C29H28ClN5O
- Molecular Weight:498.02
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT1A Receptor |
5-HT1B Receptor |
5-HT1D Receptor |
5-HT1A Receptor 8.0 (pKi) |
5-HT1B Receptor 8.1 (pKi) |
5-HT1D Receptor 8.7 (pKi) |
Chemical Information
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CAS No. 216058-27-4
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Molecular Weight 498.02
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Formula C29H28ClN5O
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SMILES
O=C(N1C2=CC(N3CCN(CC3)C)=C(C=C2CC1)Cl)NC4=C5C=CC=CC5=C(C6=CC=NC=C6)C=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
SB-272183 Related Classifications
HY-116908 Related Classifications
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