VU0631019
VU0631019 is a potent antagonist of 5-HT2B, with the IC50 of 29 nM. VU0631019 is predicted to have very limited potential for brain penetration in human subjects, as is predicted to be substrates for P-gp-mediated efflux in humans.
For research use only. We do not sell to patients.
- CAS No.: 1235656-95-7
- Formula: C20H26ClN3O2
- Molecular Weight:375.89
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
More
Biological Activity
|
5-HT2B Receptor |
5-HT2B Receptor 29 nM (IC50) |
Chemical Information
-
CAS No. 1235656-95-7
-
Molecular Weight 375.89
-
Formula C20H26ClN3O2
-
SMILES
O=C(NCC1CCN(CC1)CC2=C(C)OC(C)=C2)NC3=C(Cl)C=CC=C3
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)